Activity record

PGDB_A007899

Assay: % DegradationQC: ambiguous
Activity overview

DC50 <= 50 nM

Cell lineJurkat
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS002078
PatentCN121698875A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C024776
Compound IDPGDB_C024776
Compound782;782;化合物782
Source record IDPGDB_C024776
InChIKeyPZWBQBCCZDNZFV-FIBGUPNXSA-N

Assay context

Assay IDPGDB_AS002078
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Detection targetprotein_degradation
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens

Source evidence

Patent IDCN121698875A
Compound location

782;782;化合物782

782;782;化合物782 enlarged structure782;782;化合物782 location on patent page 41
Activity table
Page 396 · table single