Activity record

PGDB_A008885

Assay: biochemicalTarget: CRBNQC: standardized
Activity overview

IC50 > 1000 nM

TargetCRBN
E3 ligaseCRBN
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS000712
PatentWO2022219407A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009973
Compound IDPGDB_C009973
Compound72
Source record IDPGDB_C009973
InChIKeyAMCKRIRQIBKIDA-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000712
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
TargetCRBN
E3CRBN

Source evidence

Patent IDWO2022219407A1
Compound location

72

72 enlarged structure72 location on patent page 122
Activity table
Page 185 · table single