Activity record

PGDB_A016930

Assay: % DegradationQC: ambiguous
Activity overview

DC50 <= 50 nM

Cell lineJurkat
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS002078
PatentCN121698875A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C024819
Compound IDPGDB_C024819
Compound1070;1070;化合物1070
Source record IDPGDB_C024819
InChIKeyXPVQKSMJDLQRJZ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002078
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Detection targetprotein_degradation
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens

Source evidence

Patent IDCN121698875A
Compound location

1070;1070;化合物1070

1070;1070;化合物1070 enlarged structure1070;1070;化合物1070 location on patent page 49
Activity table
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