Activity record

PGDB_A046846

Assay: % DegradationQC: ambiguous
Activity overview

DC50 = 50-500 nM

Cell lineJurkat
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS002078
PatentCN121698875A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C024752
Compound IDPGDB_C024752
Compound87;87;87
Source record IDPGDB_C024752
InChIKeyBHDWZHAKRLXBKP-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002078
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Detection targetprotein_degradation
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens

Source evidence

Patent IDCN121698875A
Compound location

87;87;87

87;87;87 enlarged structure87;87;87 location on patent page 21
Activity table
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