Activity record

PGDB_A059269

Assay: biochemicalTarget: CRBNQC: standardized
Activity overview

IC50 = 100-1000 nM

TargetCRBN
E3 ligaseCRBN
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS000712
PatentWO2022219407A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009968
Compound IDPGDB_C009968
Compound71
Source record IDPGDB_C009968
InChIKeyYHAOJUVJIQSFRU-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000712
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
TargetCRBN
E3CRBN

Source evidence

Patent IDWO2022219407A1
Compound location

71

71 enlarged structure71 location on patent page 122
Activity table
Page 185 · table single