Activity record

PGDB_A075260

Assay: % DegradationQC: ambiguous
Activity overview

DC50 <= 50 nM

Cell lineJurkat
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS002078
PatentCN121698875A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C024741
Compound IDPGDB_C024741
Compound303;303;化合物303
Source record IDPGDB_C024741
InChIKeyZTGKHTHHPFWGPM-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002078
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Detection targetprotein_degradation
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens

Source evidence

Patent IDCN121698875A
Compound location

303;303;化合物303

303;303;化合物303 enlarged structure303;303;化合物303 location on patent page 28
Activity table
Page 396 · table single