PatGlueDB | Molecular Glue Patent Bioactivity Database

Patent summary

Publication numberAR127239A1

AssigneePeloton Therapeutics

TitleSULTAMAS AND TRICYCLIC SULFAMIDES AS ANTI-TUMORAL AGENTS

Family ID85988823

Family members6

Filing year2022

Publication date2024-01-03

JurisdictionAR

Compounds100

Activity records279

Assays3

Activity compounds and values

Activity records

279 records

	Control		Value		Concentration	Time				Record ID	Compound	Assay	Details
EC50	-	=	0.0026	uM	-	—	RBM39	DCAF15	-	PGDB_A008133	PGDB_C005605	PGDB_AS002536	View
EC50	-	=	0.0031	uM	-	—	RBM39	DCAF15	-	PGDB_A008138	PGDB_C005555	PGDB_AS002536	View
IC50	-	=	1.0678	uM	-	—	DCAF15	DCAF15	-	PGDB_A008577	PGDB_C005569	PGDB_AS000201	View
EC50	-	=	0.0011	uM	-	—	RBM39	DCAF15	-	PGDB_A008990	PGDB_C005599	PGDB_AS002536	View
IC50	-	=	1.791	uM	-	—	RBM39	-	HCT116	PGDB_A009052	PGDB_C005633	PGDB_AS002257	View
EC50	-	=	0.0007	uM	-	—	RBM39	DCAF15	-	PGDB_A009083	PGDB_C005627	PGDB_AS002536	View
EC50	-	=	0.0177	uM	-	—	RBM39	DCAF15	-	PGDB_A010054	PGDB_C005630	PGDB_AS002536	View
IC50	-	=	19.953	uM	-	—	DCAF15	DCAF15	-	PGDB_A010065	PGDB_C005554	PGDB_AS000201	View
EC50	-	=	0.2121	uM	-	—	RBM39	DCAF15	-	PGDB_A010317	PGDB_C005648	PGDB_AS002536	View
IC50	-	=	0.1257	uM	-	—	RBM39	-	HCT116	PGDB_A010379	PGDB_C005583	PGDB_AS002257	View
IC50	-	=	52.219	uM	-	—	DCAF15	DCAF15	-	PGDB_A010637	PGDB_C005574	PGDB_AS000201	View
EC50	-	=	0.0016	uM	-	—	RBM39	DCAF15	-	PGDB_A010891	PGDB_C005642	PGDB_AS002536	View
IC50	-	=	3.1602	uM	-	—	RBM39	-	HCT116	PGDB_A011726	PGDB_C005557	PGDB_AS002257	View
IC50	-	=	0.3513	uM	-	—	RBM39	-	HCT116	PGDB_A011735	PGDB_C005612	PGDB_AS002257	View
EC50	-	=	0.004	uM	-	—	RBM39	DCAF15	-	PGDB_A011874	PGDB_C005584	PGDB_AS002536	View
IC50	-	=	0.4146	uM	-	—	RBM39	-	HCT116	PGDB_A012296	PGDB_C005570	PGDB_AS002257	View
IC50	-	=	100	uM	-	—	DCAF15	DCAF15	-	PGDB_A012304	PGDB_C005559	PGDB_AS000201	View
IC50	-	=	0.5799	uM	-	—	DCAF15	DCAF15	-	PGDB_A012361	PGDB_C005601	PGDB_AS000201	View
IC50	-	=	5	uM	-	—	RBM39	-	HCT116	PGDB_A012439	PGDB_C005607	PGDB_AS002257	View
IC50	-	=	0.0518	uM	-	—	DCAF15	DCAF15	-	PGDB_A012701	PGDB_C005640	PGDB_AS000201	View

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