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SIMM · NJU
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SIMM · NJU
Patent
EP4573088A1
132 compounds
133 activity records
1 assays
Patent summary
Publication number
EP4573088A1
Assignee
Recursion Pharmaceuticals
Title
Heterocycle rbm39 modulators
Family ID
88018171
Family members
12
Family patent IDs
AU2023324686A1
CA3261302A1
CL2025000421A1
CN119630658A
CO2025000357A2
EP4573088A1
IL318189A
JP2025529797A
KR20250048008A
MX2025001802A
US20240092770A1
WO2024039689A1
Filing year
2023
Publication date
2025-06-25
Jurisdiction
EP
Compounds
132
Activity records
133
Assays
1
Activity compounds and values
Activity records
133 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
EC50
-
=
353.8
nM
-
—
RBM39
DCAF15
-
PGDB_A007098
PGDB_C007602
PGDB_AS000315
View
EC50
-
=
4190.8
nM
-
—
RBM39
DCAF15
-
PGDB_A007935
PGDB_C007604
PGDB_AS000315
View
EC50
-
=
3262.1
nM
-
—
RBM39
DCAF15
-
PGDB_A008563
PGDB_C007666
PGDB_AS000315
View
EC50
-
=
420.7
nM
-
—
RBM39
DCAF15
-
PGDB_A009620
PGDB_C007628
PGDB_AS000315
View
EC50
-
=
738.2
nM
-
—
RBM39
DCAF15
-
PGDB_A009701
PGDB_C007632
PGDB_AS000315
View
EC50
-
=
1167.5
nM
-
—
RBM39
DCAF15
-
PGDB_A010090
PGDB_C007623
PGDB_AS000315
View
EC50
-
=
1972.3
nM
-
—
RBM39
DCAF15
-
PGDB_A010165
PGDB_C007661
PGDB_AS000315
View
EC50
-
=
99.6
nM
-
—
RBM39
DCAF15
-
PGDB_A010175
PGDB_C007668
PGDB_AS000315
View
EC50
-
=
916.8
nM
-
—
RBM39
DCAF15
-
PGDB_A012528
PGDB_C007671
PGDB_AS000315
View
EC50
-
=
1633.8
nM
-
—
RBM39
DCAF15
-
PGDB_A012967
PGDB_C007589
PGDB_AS000315
View
EC50
-
=
1619.6
nM
-
—
RBM39
DCAF15
-
PGDB_A013967
PGDB_C007665
PGDB_AS000315
View
EC50
-
=
241.1
nM
-
—
RBM39
DCAF15
-
PGDB_A014510
PGDB_C007713
PGDB_AS000315
View
EC50
-
=
2069.1
nM
-
—
RBM39
DCAF15
-
PGDB_A016279
PGDB_C007662
PGDB_AS000315
View
EC50
-
=
978.2
nM
-
—
RBM39
DCAF15
-
PGDB_A016421
PGDB_C007703
PGDB_AS000315
View
EC50
-
=
104.3
nM
-
—
RBM39
DCAF15
-
PGDB_A016687
PGDB_C007651
PGDB_AS000315
View
EC50
-
=
2070.6
nM
-
—
RBM39
DCAF15
-
PGDB_A017304
PGDB_C007644
PGDB_AS000315
View
EC50
-
=
55.2
nM
-
—
RBM39
DCAF15
-
PGDB_A017405
PGDB_C007608
PGDB_AS000315
View
EC50
-
=
391.3
nM
-
—
RBM39
DCAF15
-
PGDB_A017713
PGDB_C007712
PGDB_AS000315
View
EC50
-
=
649.9
nM
-
—
RBM39
DCAF15
-
PGDB_A018828
PGDB_C007675
PGDB_AS000315
View
EC50
-
=
207
nM
-
—
RBM39
DCAF15
-
PGDB_A019822
PGDB_C007711
PGDB_AS000315
View