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SIMM · NJU
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SIMM · NJU
Patent
WO2021239117A1
184 compounds
184 activity records
3 assays
Patent summary
Publication number
WO2021239117A1
Assignee
Cullgen Shanghai
Title
Modified proteins and protein degraders
Family ID
78722770
Family members
8
Family patent IDs
CN116472292A
EP4157888A1
EP4157888A4
JP2023529099A
JPWO2021239117A5
US20230057177A1
US20240066136A1
WO2021239117A1
Filing year
2021
Publication date
2021-12-02
Jurisdiction
WO
Compounds
184
Activity records
184
Assays
3
Activity compounds and values
Activity records
184 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
Kd
-
<
20
uM
-
—
DDB1
-
-
PGDB_A007188
PGDB_C009391
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A007301
PGDB_C009303
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A007815
PGDB_C009422
PGDB_AS000435
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A007986
PGDB_C009363
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A008931
PGDB_C009370
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A009066
PGDB_C009380
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A009254
PGDB_C009369
PGDB_AS002280
View
Kd
-
<
20
uM
-
—
DDB1
-
-
PGDB_A009525
PGDB_C009315
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A009717
PGDB_C009277
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A010727
PGDB_C009404
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A011294
PGDB_C009371
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A011566
PGDB_C009400
PGDB_AS002280
View
Kd
-
>
100
uM
-
—
DDB1
-
-
PGDB_A011840
PGDB_C009392
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A011937
PGDB_C009393
PGDB_AS002280
View
Kd
-
<
20
uM
-
—
DDB1
-
-
PGDB_A012262
PGDB_C009442
PGDB_AS000915
View
Kd
-
<
20
uM
-
—
DDB1
-
-
PGDB_A012889
PGDB_C009456
PGDB_AS000915
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A013449
PGDB_C009299
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A013629
PGDB_C009331
PGDB_AS002280
View
Kd
-
<
20
uM
-
—
DDB1
-
-
PGDB_A013901
PGDB_C009376
PGDB_AS002280
View
Kd
-
=
20-100
uM
-
—
DDB1
-
-
PGDB_A013958
PGDB_C009382
PGDB_AS002280
View