PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Loading patent
Loading detail record from the SQLite release...
PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Patent
WO2023059899A1
39 compounds
72 activity records
3 assays
Patent summary
Publication number
WO2023059899A1
Assignee
Triana Biomedicines
Title
Fused bicyclic substituted n-(1h-indol-7-yl)benzenesulfonamides and uses thereof
Family ID
84329416
Family members
2
Family patent IDs
US20240425486A1
WO2023059899A1
Filing year
2022
Publication date
2023-04-13
Jurisdiction
WO
Compounds
39
Activity records
72
Assays
3
Activity compounds and values
Activity records
72 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
EC50
-
<=
100
uM
-
—
RBM39
DCAF15
-
PGDB_A007124
PGDB_C010022
PGDB_AS001283
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A007464
PGDB_C010018
PGDB_AS002163
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A007773
PGDB_C010013
PGDB_AS002163
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A008104
PGDB_C010029
PGDB_AS002163
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
PGDB_A008442
PGDB_C010016
PGDB_AS001283
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A008848
PGDB_C010028
PGDB_AS002163
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
PGDB_A009262
PGDB_C010009
PGDB_AS001283
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A009344
PGDB_C010010
PGDB_AS002163
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
PGDB_A009792
PGDB_C010003
PGDB_AS001283
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
PGDB_A009999
PGDB_C010015
PGDB_AS001283
View
IC50
-
<=
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A010556
PGDB_C010023
PGDB_AS002163
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A012450
PGDB_C010030
PGDB_AS002163
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
PGDB_A013745
PGDB_C010006
PGDB_AS001283
View
IC50
-
<=
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A016902
PGDB_C010015
PGDB_AS002163
View
IC50
-
>
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A018028
PGDB_C010020
PGDB_AS002163
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
PGDB_A018461
PGDB_C010026
PGDB_AS001283
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
PGDB_A018552
PGDB_C010007
PGDB_AS001283
View
EC50
-
<=
1
uM
-
—
RBM39
DCAF15
-
PGDB_A020143
PGDB_C010018
PGDB_AS001283
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
PGDB_A020493
PGDB_C010024
PGDB_AS001283
View
EC50
-
<=
10
uM
-
—
RBM39
DCAF15
-
PGDB_A021680
PGDB_C010010
PGDB_AS001283
View