PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Loading patent
Loading detail record from the SQLite release...
PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Patent
WO2023274246A1
132 compounds
145 activity records
2 assays
Patent summary
Publication number
WO2023274246A1
Assignee
Chengdu Fendi Pharmaceutical
Title
Amide compound and use thereof
Family ID
84690387
Family members
6
Family patent IDs
CN117440948A
EP4365170A1
EP4365170A4
JP2024524765A
US20240368113A1
WO2023274246A1
Filing year
2022
Publication date
2024-05-08
Jurisdiction
WO
Compounds
132
Activity records
145
Assays
2
Activity compounds and values
Activity records
145 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A007033
PGDB_C002321
PGDB_AS002583
View
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A007767
PGDB_C002430
PGDB_AS002583
View
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A008328
PGDB_C002316
PGDB_AS002583
View
IC50
-
=
1-10
nM
-
—
-
-
MV-4-11
PGDB_A008374
PGDB_C002443
PGDB_AS002583
View
IC50
-
=
1-10
nM
-
—
-
-
MV-4-11
PGDB_A008425
PGDB_C002363
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A010589
PGDB_C002440
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A010805
PGDB_C002336
PGDB_AS002583
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A010937
PGDB_C002381
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A011912
PGDB_C002391
PGDB_AS002583
View
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A012009
PGDB_C002334
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A012400
PGDB_C002413
PGDB_AS002583
View
IC50
-
=
1-10
nM
-
—
-
-
MV-4-11
PGDB_A013065
PGDB_C002401
PGDB_AS002583
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A014588
PGDB_C002393
PGDB_AS002583
View
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A016069
PGDB_C002369
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A016384
PGDB_C002335
PGDB_AS002583
View
IC50
-
=
1-10
nM
-
—
-
-
MV-4-11
PGDB_A016987
PGDB_C002424
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A018145
PGDB_C002356
PGDB_AS002583
View
IC50
-
<
1
nM
-
—
-
-
MV-4-11
PGDB_A018584
PGDB_C002365
PGDB_AS002583
View
IC50
-
>
100
nM
-
—
-
-
MV-4-11
PGDB_A018698
PGDB_C002388
PGDB_AS002583
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A019509
PGDB_C002330
PGDB_AS002583
View