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SIMM · NJU
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SIMM · NJU
Patent
WO2025189015A1
47 compounds
47 activity records
1 assays
Patent summary
Publication number
WO2025189015A1
Assignee
Seed Therapeutics
Title
Heteroaromatic indolesulfonamides
Family ID
96991643
Family members
2
Family patent IDs
WO2025189015A1
WO2025189015A8
Filing year
2025
Publication date
2025-09-12
Jurisdiction
WO
Compounds
47
Activity records
47
Assays
1
Activity compounds and values
Activity records
47 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A007043
PGDB_C027673
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A008800
PGDB_C027671
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A009683
PGDB_C027686
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A012514
PGDB_C027646
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A015117
PGDB_C027670
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A015331
PGDB_C027683
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A021221
PGDB_C027652
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A022510
PGDB_C027649
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A026237
PGDB_C027667
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A026757
PGDB_C027687
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A027608
PGDB_C027661
PGDB_AS000963
View
IC50
-
<
500
nM
-
—
RBM39
-
HCT116
PGDB_A027648
PGDB_C027647
PGDB_AS000963
View
IC50
-
<
500
nM
-
—
RBM39
-
HCT116
PGDB_A028528
PGDB_C027689
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A029761
PGDB_C027677
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A030886
PGDB_C027656
PGDB_AS000963
View
IC50
-
<
500
nM
-
—
RBM39
-
HCT116
PGDB_A031306
PGDB_C027648
PGDB_AS000963
View
IC50
-
>
1000
nM
-
—
RBM39
-
HCT116
PGDB_A031562
PGDB_C027669
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A031783
PGDB_C007711
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A032152
PGDB_C027645
PGDB_AS000963
View
IC50
-
=
500-1000
nM
-
—
RBM39
-
HCT116
PGDB_A032624
PGDB_C027678
PGDB_AS000963
View