Activity record

PGDB_A000257

Assay: viabilityTarget: ARQC: standardized
Activity overview

IC50 = 0.053 nM

TargetAR
Cell lineVCaP
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000271
PatentWO2026061104A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C029768
Compound IDPGDB_C029768
CompoundAR-P-241
Source record IDPGDB_C029768
InChIKeyIPZBJXXOIDSREW-XQLHXAQRSA-N

Assay context

Assay IDPGDB_AS000271
Assay familyviability
Assay systemcell_based
ReadoutIC50
Detection target% Cell viability
TargetAR
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2026061104A1
Compound location

AR-P-241

AR-P-241 enlarged structureAR-P-241 location on patent page 186
Activity table
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