Activity record

PGDB_A001641

Assay: viabilityTarget: ARQC: standardized
Activity overview

IC50 = 0.065 nM

TargetAR
Cell lineVCaP
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000271
PatentWO2026061104A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C030090
Compound IDPGDB_C030090
CompoundAR-P-221
Source record IDPGDB_C030090
InChIKeyALCJRHQAPGIYKB-UFNASBJGSA-N

Assay context

Assay IDPGDB_AS000271
Assay familyviability
Assay systemcell_based
ReadoutIC50
Detection target% Cell viability
TargetAR
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2026061104A1
Compound location

AR-P-221

AR-P-221 enlarged structureAR-P-221 location on patent page 179
Activity table
Page 272 · table start
Page 273 · table middle
Page 274 · table end