Activity record

PGDB_A002835

Assay: % DegradationTarget: VAV1QC: standardized
Activity overview

Dmax = 98.7 %

TargetVAV1
Cell lineJurkat
Time24 h
Assay / Readoutluminescence / Dmax
Assay IDPGDB_AS001360
PatentWO2026098637A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C031197
Compound IDPGDB_C031197
Compound4
Source record IDPGDB_C031197
InChIKeyVSJTUBBPTOHBIL-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001360
Assay family% Degradation
Assay systemcell_based
ReadoutDmax
Technologyluminescence
Treatment time24 h
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens

Source evidence

Patent IDWO2026098637A1
Compound location

4

4 enlarged structure4 location on patent page 121
Activity table
Page 98 · table single