Activity record

PGDB_A007955

Assay: % DegradationTarget: GSPT1QC: standardized
Activity overview

DC50 = 16 nM

TargetGSPT1
Cell lineABC-1
Time6 h
Assay / Readoutfluorescence / DC50
Assay IDPGDB_AS001474
PatentCN119264113A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000673
Compound IDPGDB_C000673
Compound化合物 3;化合物 3;化合物3
Source record IDPGDB_C000673
InChIKeyCWHJQFPZRKGIHE-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001474
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Technologyfluorescence
Treatment time6 h
TargetGSPT1
E3Not specified
Cell lineABC-1
OrganismHomo sapiens

Source evidence

Patent IDCN119264113A
Compound location

化合物 3;化合物 3;化合物3

化合物 3;化合物 3;化合物3 enlarged structure化合物 3;化合物 3;化合物3 location on patent page 4
Activity table
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