Activity record

PGDB_A010512

Assay: biochemicalTarget: DCAF15QC: standardized
Activity overview

IC50 < 100 uM

TargetDCAF15
E3 ligaseDCAF15
Time1 h
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS000694
PatentWO2022173805A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009789
Compound IDPGDB_C009789
Compound233.0
Source record IDPGDB_C009789
InChIKeyTWRRGMJCDXYSSK-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000694
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
Treatment time1 h
TargetDCAF15
E3DCAF15

Source evidence

Patent IDWO2022173805A1
Compound location

233.0

233.0 enlarged structure233.0 location on patent page 166
Activity table
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