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SIMM · NJU
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SIMM · NJU
Patent
WO2022173805A1
173 compounds
353 activity records
4 assays
Patent summary
Publication number
WO2022173805A1
Assignee
Triana Biomedicines
Title
Amide and ether substituted n-(1h-indol-7-yl)benzenesulfonamides and uses thereof
Family ID
80623491
Family members
2
Family patent IDs
US20240327351A1
WO2022173805A1
Filing year
2022
Publication date
2022-08-18
Jurisdiction
WO
Compounds
173
Activity records
353
Assays
4
Activity compounds and values
Activity records
353 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
PGDB_A007146
PGDB_C009790
PGDB_AS000136
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A007578
PGDB_C009660
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A007643
PGDB_C009663
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A007796
PGDB_C009705
PGDB_AS000694
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
PGDB_A008240
PGDB_C009647
PGDB_AS000136
View
IC50
-
>
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A008673
PGDB_C009765
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A008698
PGDB_C009625
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A008822
PGDB_C009792
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A008881
PGDB_C009658
PGDB_AS000694
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
PGDB_A008923
PGDB_C009677
PGDB_AS000136
View
IC50
-
>
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A009270
PGDB_C009752
PGDB_AS000694
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
PGDB_A009492
PGDB_C009646
PGDB_AS000136
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A009947
PGDB_C009673
PGDB_AS000694
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
PGDB_A010300
PGDB_C009654
PGDB_AS000136
View
IC50
-
<
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A010512
PGDB_C009789
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A010761
PGDB_C009656
PGDB_AS000694
View
IC50
-
>
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A010803
PGDB_C009745
PGDB_AS000694
View
IC50
-
<
10
uM
-
—
DCAF15
DCAF15
-
PGDB_A010824
PGDB_C009766
PGDB_AS000694
View
IC50
-
>
100
uM
-
—
DCAF15
DCAF15
-
PGDB_A011130
PGDB_C009788
PGDB_AS000694
View
EC50
-
<
100
uM
-
—
RBM39
DCAF15
-
PGDB_A011204
PGDB_C009735
PGDB_AS000136
View