Activity record

PGDB_A013406

Assay: % DegradationTarget: ERQC: standardized
Activity overview

IC50 = 0.4 nM

TargetER
Cell lineLNCaP
Time6 d
Assay / Readoutluminescence / IC50
Assay IDPGDB_AS001923
PatentCN118984820A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006923
Compound IDPGDB_C006923
CompoundC2;C2
Source record IDPGDB_C006923
InChIKeyHMUJPMUPBWROPO-VWLOTQADSA-N

Assay context

Assay IDPGDB_AS001923
Assay family% Degradation
Assay systemcell_based
ReadoutIC50
Technologyluminescence
Treatment time6 d
TargetER
E3Not specified
Cell lineLNCaP

Source evidence

Patent IDCN118984820A
Compound location

C2;C2

C2;C2 enlarged structureC2;C2 location on patent page 106
Activity table
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