Activity record

PGDB_A021762

Assay: cellular_functionTarget: BLOC1S6QC: ambiguous
Activity overview

EC50 = 1.22 uM

TargetBLOC1S6
Cell lineHEK293T
Time24 h
Assay / Readoutfluorescence / EC50
Assay IDPGDB_AS002050
PatentJP2024545831A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C008307
Compound IDPGDB_C008307
CompoundC10
Source record IDPGDB_C008307
InChIKeyAAVSZQDNLAZAOL-KBRGNYCBSA-N

Assay context

Assay IDPGDB_AS002050
Assay familycellular_function
Assay systemcell_based
ReadoutEC50
Technologyfluorescence
Treatment time24 h
TargetBLOC1S6
E3Not specified
Cell lineHEK293T
OrganismHomo sapiens

Source evidence

Patent IDJP2024545831A
Compound location

C10

C10 enlarged structureC10 location on patent page 27
Activity table
Page 29 · table single