PatGlueDB | Molecular Glue Patent Bioactivity Database

Patent summary

Publication numberJP2024545831A

AssigneeInstitute of Medicinal Biotechnology, CAMS & PUMC

TitlePerinaphthenone compounds and their uses

Family ID78490979

Family members6

Filing year2022

Publication date2024-12-13

JurisdictionJP

Compounds15

Activity records44

Assays3

Activity compounds and values

Activity records

44 records

	Control		Value		Concentration	Time				Record ID	Compound	Assay	Details
EC50	-	=	27.85	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A008434	PGDB_C008304	PGDB_AS002050	View
EC50	-	=	0.88	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A008589	PGDB_C008307	PGDB_AS002145	View
EC50	-	=	1.14	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A014449	PGDB_C008299	PGDB_AS002145	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A014802	PGDB_C008306	PGDB_AS001447	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A016530	PGDB_C008307	PGDB_AS001447	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A018938	PGDB_C008298	PGDB_AS001447	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A019225	PGDB_C008302	PGDB_AS001447	View
EC50	-	=	0.92	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A019604	PGDB_C008309	PGDB_AS002050	View
EC50	-	=	1.22	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A021762	PGDB_C008307	PGDB_AS002050	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A021887	PGDB_C008311	PGDB_AS001447	View
EC50	-	=	0.55	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A024237	PGDB_C008305	PGDB_AS002050	View
EC50	-	=	2.09	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A024374	PGDB_C008302	PGDB_AS002145	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A025667	PGDB_C008309	PGDB_AS001447	View
EC50	-	=	2.22	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A027459	PGDB_C008302	PGDB_AS002050	View
EC50	-	=	0.58	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A028847	PGDB_C008298	PGDB_AS002050	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A029126	PGDB_C008301	PGDB_AS001447	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A033885	PGDB_C008300	PGDB_AS001447	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A034299	PGDB_C008305	PGDB_AS001447	View
EC50	-	=	1.25	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A035574	PGDB_C008300	PGDB_AS002050	View
CC50	-	>	100	uM	-	—	BLOC1S6	-	HEK293T	PGDB_A037590	PGDB_C008308	PGDB_AS001447	View

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