Activity record

PGDB_A027467

Assay: % DegradationTarget: CDK13QC: ambiguous
Activity overview

IC50 <= 0.1 uM

TargetCDK13
Assay / ReadoutIC50 / % Degradation
Assay IDPGDB_AS001146
PatentWO2025110815A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C011002
Compound IDPGDB_C011002
Compound115.0
Source record IDPGDB_C011002
InChIKeyHKHCDZAAXKYDBN-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001146
Assay family% Degradation
Assay systemcell_based
ReadoutIC50
TargetCDK13
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

115.0

115.0 enlarged structure115.0 location on patent page 136
Activity table
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