Activity record

PGDB_A030565

Assay: % DegradationTarget: CCNKQC: ambiguous
Activity overview

DC50 < 500 nM

TargetCCNK
Time24 h
Assay / Readoutluminescence / DC50
Assay IDPGDB_AS001864
PatentWO2025245472A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C012043
Compound IDPGDB_C012043
Compound181
Source record IDPGDB_C012043
InChIKeyTYFBJCHEZZWFFP-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001864
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Technologyluminescence
Treatment time24 h
Detection targetprotein_degradation
TargetCCNK
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDWO2025245472A1
Compound location

181

181 enlarged structure181 location on patent page 80
Activity table
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