Activity record

PGDB_A034075

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

IC50 = 10-50 uM

TargetGSPT1
E3 ligaseCRBN
Cell lineKG-1
Time72 h
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS001194
PatentCN118234721A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C019833
Compound IDPGDB_C019833
Compound比较化合物 1
Source record IDPGDB_C001245
InChIKeyOCPDIVVLRZPTOE-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001194
Assay familyviability
Assay systemcell_based
ReadoutIC50
Treatment time72 h
TargetGSPT1
E3CRBN
Cell lineKG-1

Source evidence

Patent IDCN118234721A
Compound location

比较化合物 1

比较化合物 1 enlarged structure比较化合物 1 location on patent page 61
Activity table
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