Activity record

PGDB_A035851

Assay: bindingTarget: VHLQC: ambiguous
Activity overview

Ki < 300 nM

TargetVHL
E3 ligaseVHL
Time1 h
Assay / Readoutfluorescence / Ki
Assay IDPGDB_AS000103
PatentCN119613482A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006931
Compound IDPGDB_C006931
CompoundI-8;I-8
Source record IDPGDB_C006931
InChIKeyNUQLYOLPZZCKRU-TVZXLZGTSA-N

Assay context

Assay IDPGDB_AS000103
Assay familybinding
Assay systembiochemical
ReadoutKi
Technologyfluorescence
Treatment time1 h
TargetVHL | ELOB | ELOC
E3VHL | ELOB | ELOC

Source evidence

Patent IDCN119613482A
Compound location

I-8;I-8

I-8;I-8 enlarged structureI-8;I-8 location on patent page 3
Activity table
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