Activity record

PGDB_A036025

Assay: % DegradationTarget: ESR1QC: ambiguous
Activity overview

degradation = 85 %

TargetESR1
Cell lineMCF-7
Concentration0.3 uM
Time4 h
Assay / Readout% Degradation
Assay IDPGDB_AS001441
PatentCN118984820A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006885
Compound IDPGDB_C006885
Compound3
Source record IDPGDB_C006885
InChIKeyAWHNYVYKKLSGAQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001441
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration0.3 uM
Treatment time4 h
TargetESR1
E3Not specified
Cell lineMCF-7

Source evidence

Patent IDCN118984820A
Compound location

3

3 enlarged structure3 location on patent page 40
Activity table
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