Activity record

PGDB_A036751

Assay: biochemicalTarget: NFE2L2QC: standardized
Activity overview

EC50 < 1 uM

TargetNFE2L2
E3 ligaseBTRC | FBXW11
Time1 h
Assay / ReadoutEC50 / biochemical
Assay IDPGDB_AS001397
PatentWO2025179005A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C021135
Compound IDPGDB_C021135
Compound217
Source record IDPGDB_C021135
InChIKeyCMVJBOGQAGCLQK-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001397
Assay familybiochemical
Assay systembiochemical
ReadoutEC50
Treatment time1 h
TargetNFE2L2
E3BTRC | FBXW11 | SKP1

Source evidence

Patent IDWO2025179005A1
Compound location

217

217 enlarged structure217 location on patent page 509
Activity table
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