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SIMM · NJU
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SIMM · NJU
Patent
WO2025179005A1
349 compounds
685 activity records
6 assays
Patent summary
Publication number
WO2025179005A1
Assignee
Triana Biomedicines
Title
Molecular glues and uses thereof
Family ID
94974206
Family members
1
Family patent IDs
WO2025179005A1
Filing year
2025
Publication date
2025-08-28
Jurisdiction
WO
Compounds
349
Activity records
685
Assays
6
Activity compounds and values
Activity records
685 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A007219
PGDB_C020796
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A007293
PGDB_C020826
PGDB_AS000440
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A007325
PGDB_C021106
PGDB_AS002352
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A007347
PGDB_C021012
PGDB_AS001171
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A007571
PGDB_C020816
PGDB_AS002080
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A007599
PGDB_C020863
PGDB_AS000440
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A007685
PGDB_C020830
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A007958
PGDB_C020870
PGDB_AS000440
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A007991
PGDB_C021115
PGDB_AS002352
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A008167
PGDB_C021088
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A008437
PGDB_C021074
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A008604
PGDB_C021048
PGDB_AS002352
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A008781
PGDB_C020894
PGDB_AS002080
View
EC50
-
>
10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A008997
PGDB_C021016
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A009070
PGDB_C021017
PGDB_AS001171
View
EC50
-
=
1-10
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A009142
PGDB_C020907
PGDB_AS002080
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A009182
PGDB_C021142
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A009245
PGDB_C021027
PGDB_AS002352
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
PGDB_A009364
PGDB_C021105
PGDB_AS002352
View
EC50
-
<
1
uM
-
—
NFE2L2
BTRC | FBXW11
-
PGDB_A009672
PGDB_C020826
PGDB_AS002080
View