Activity record

PGDB_A037341

Assay: biochemicalTarget: RBM39QC: ambiguous
Activity overview

EC50 = 429.1 nM

TargetRBM39
E3 ligaseDCAF15
Time60 min
Assay / ReadoutEC50 / biochemical
Assay IDPGDB_AS000315
PatentEP4573088A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C007589
Compound IDPGDB_C007589
CompoundExample 3
Source record IDPGDB_C007589
InChIKeySXHLKLVJZNTBQG-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000315
Assay familybiochemical
Assay systembiochemical
ReadoutEC50
Treatment time60 min
TargetRBM39
E3DCAF15 | DDA1 | DDB1

Source evidence

Patent IDEP4573088A1
Compound location

Example 3

Example 3 enlarged structureExample 3 location on patent page 99
Activity table
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