Activity record

PGDB_A039460

Assay: % DegradationTarget: IKZF2QC: standardized
Activity overview

DC50 = 0.043 uM

TargetIKZF2
Cell lineMOLT-4
Time6 h
Assay / Readoutluminescence / DC50
Assay IDPGDB_AS000536
PatentCA3215907A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006102
Compound IDPGDB_C006102
Compound146;146
Source record IDPGDB_C006102
InChIKeyWMUQHLIIVQBYHB-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000536
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Technologyluminescence
Treatment time6 h
TargetIKZF2
E3Not specified
Cell lineMOLT-4

Source evidence

Patent IDCA3215907A1
Compound location

146;146

146;146 enlarged structure146;146 location on patent page 65
Activity table
Page 98 · table start
Page 99 · table end