Activity record

PGDB_A040414

Assay: % DegradationTarget: GSPT1QC: standardized
Activity overview

DC50 > 30 uM

TargetGSPT1
Cell lineHEK293T
Time24 h
Assay / Readoutluminescence / DC50
Assay IDPGDB_AS002212
PatentAR126418A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000472
Compound IDPGDB_C000472
Compound134;134
Source record IDPGDB_C000472
InChIKeyHOOUEZZAUDFDOC-PFIFLBKHSA-N

Assay context

Assay IDPGDB_AS002212
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Technologyluminescence
Treatment time24 h
TargetGSPT1
E3Not specified
Cell lineHEK293T

Source evidence

Patent IDAR126418A1
Compound location

134;134

134;134 enlarged structure134;134 location on patent page 62
Activity table
Page 187 · table start
Page 188 · table end