Activity record

PGDB_A042085

Assay: ternary_complexTarget: RBM39QC: ambiguous
Activity overview

EC50 = 0.011 uM

TargetRBM39
E3 ligaseDCAF15
Timeovernight
Assay / ReadoutEC50 / ternary_complex
Assay IDPGDB_AS002536
PatentAR127239A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C005554
Compound IDPGDB_C005554
Compound5.0
Source record IDPGDB_C005554
InChIKeyXZIRGIBFSXKDNT-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002536
Assay familyternary_complex
Assay systembiochemical
ReadoutEC50
Treatment timeovernight
TargetRBM39
E3DCAF15
OrganismHomo sapiens

Source evidence

Patent IDAR127239A1
Compound location

5.0

multi-compoundsneed check
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