Activity record

PGDB_A046056

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

DC50 > 200 nM

TargetGSPT1
Assay / ReadoutDC50 / % Degradation
Assay IDPGDB_AS001361
PatentCN120441535A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C001528
Compound IDPGDB_C001528
Compound5;化合物5
Source record IDPGDB_C001528
InChIKeyOZRNMHRJEJPMDL-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001361
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDCN120441535A
Compound location

5;化合物5

5;化合物5 enlarged structure5;化合物5 location on patent page 53
Activity table
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