Assay

PGDB_AS001361

System: cell_basedTarget: GSPT1
Assay context summary

Assay context

13 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetGSPT1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

13 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001525
DC50-<=20nM-—GSPT1--CN120441535APGDB_A011141PGDB_C001525PGDB_AS001361View
2D structure for PGDB_C001524
DC50-<=20nM-—GSPT1--CN120441535APGDB_A016652PGDB_C001524PGDB_AS001361View
2D structure for PGDB_C001526
DC50-<=20nM-—GSPT1--CN120441535APGDB_A019321PGDB_C001526PGDB_AS001361View
2D structure for PGDB_C001533
DC50-<=20nM-—GSPT1--CN120441535APGDB_A029272PGDB_C001533PGDB_AS001361View
2D structure for PGDB_C001531
DC50-<=20nM-—GSPT1--CN120441535APGDB_A034681PGDB_C001531PGDB_AS001361View
2D structure for PGDB_C001534
DC50-<=20nM-—GSPT1--CN120441535APGDB_A042790PGDB_C001534PGDB_AS001361View
2D structure for PGDB_C001530
DC50-<=20nM-—GSPT1--CN120441535APGDB_A043928PGDB_C001530PGDB_AS001361View
2D structure for PGDB_C001528
DC50->200nM-—GSPT1--CN120441535APGDB_A046056PGDB_C001528PGDB_AS001361View
2D structure for PGDB_C001535
DC50-<=20nM-—GSPT1--CN120441535APGDB_A054039PGDB_C001535PGDB_AS001361View
2D structure for PGDB_C001532
DC50-<=20nM-—GSPT1--CN120441535APGDB_A058767PGDB_C001532PGDB_AS001361View
2D structure for PGDB_C001529
DC50->200nM-—GSPT1--CN120441535APGDB_A058955PGDB_C001529PGDB_AS001361View
2D structure for PGDB_C001536
DC50-<=20nM-—GSPT1--CN120441535APGDB_A059997PGDB_C001536PGDB_AS001361View
2D structure for PGDB_C001527
DC50-<=20nM-—GSPT1--CN120441535APGDB_A075837PGDB_C001527PGDB_AS001361View
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