Activity record

PGDB_A047260

Assay: biochemicalTarget: DCAF15QC: standardized
Activity overview

IC50 > 100 uM

TargetDCAF15
E3 ligaseDCAF15
Time1 h
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS000694
PatentWO2022173805A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009790
Compound IDPGDB_C009790
Compound234.0
Source record IDPGDB_C009790
InChIKeyXUFAVCSRLJBOJO-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000694
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
Treatment time1 h
TargetDCAF15
E3DCAF15

Source evidence

Patent IDWO2022173805A1
Compound location

234.0

234.0 enlarged structure234.0 location on patent page 166
Activity table
Page 171 · table start
Page 172 · table middle
Page 173 · table end