Activity record

PGDB_A049226

Assay: viabilityTarget: CCNKQC: ambiguous
Activity overview

GI50 > 3000 nM

TargetCCNK
Cell lineVCaP
Time144 h
Assay / Readoutluminescence / GI50
Assay IDPGDB_AS001027
PatentWO2025245472A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C012023
Compound IDPGDB_C012023
Compound158;158;158
Source record IDPGDB_C012023
InChIKeyRGWIPSJWLMLVHZ-MPYYAJLASA-N

Assay context

Assay IDPGDB_AS001027
Assay familyviability
Assay systemcell_based
ReadoutGI50
Technologyluminescence
Treatment time144 h
Detection targetprotein_degradation
TargetCCNK
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2025245472A1
Compound location

158;158;158

158;158;158 enlarged structure158;158;158 location on patent page 79
Activity table
Page 220 · table start
Page 221 · table end