Activity record

PGDB_A051045

Assay: bindingTarget: VHLQC: ambiguous
Activity overview

Ki < 300 nM

TargetVHL
E3 ligaseVHL
Time1 h
Assay / Readoutfluorescence / Ki
Assay IDPGDB_AS000103
PatentCN119613482A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006933
Compound IDPGDB_C006933
CompoundI-10;I-10
Source record IDPGDB_C006933
InChIKeyKJADOTASGIAXIH-SSEPRJSISA-N

Assay context

Assay IDPGDB_AS000103
Assay familybinding
Assay systembiochemical
ReadoutKi
Technologyfluorescence
Treatment time1 h
TargetVHL | ELOB | ELOC
E3VHL | ELOB | ELOC

Source evidence

Patent IDCN119613482A
Compound location

I-10;I-10

I-10;I-10 enlarged structureI-10;I-10 location on patent page 3
Activity table
Page 14 · table single