Activity record

PGDB_A066199

Assay: ternary_complexTarget: RBM39QC: standardized
Activity overview

EC50 <= 1 uM

TargetRBM39
E3 ligaseDCAF15
Time<= 1 uM
Assay / ReadoutAlphaLISA / EC50
Assay IDPGDB_AS001283
PatentWO2023059899A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010008
Compound IDPGDB_C010008
Compound10
Source record IDPGDB_C010008
InChIKeyBHABGTJGTWDLRN-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001283
Assay familyternary_complex
Assay systembiochemical
ReadoutEC50
TechnologyAlphaLISA
Treatment time<= 1 uM
TargetRBM39
E3DCAF15

Source evidence

Patent IDWO2023059899A1
Compound location

10

10 enlarged structure10 location on patent page 24
Activity table
Page 55 · table start
Page 56 · table end