Activity record

PGDB_A066225

Assay: % DegradationTarget: IKZF2QC: standardized
Activity overview

DC50 = 0.022 uM

TargetIKZF2
Cell lineMOLT-4
Time6 h
Assay / Readoutluminescence / DC50
Assay IDPGDB_AS000536
PatentCA3215907A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006105
Compound IDPGDB_C006105
Compound149;149;149
Source record IDPGDB_C006105
InChIKeyHEIOPGMVMLJGPO-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000536
Assay family% Degradation
Assay systemcell_based
ReadoutDC50
Technologyluminescence
Treatment time6 h
TargetIKZF2
E3Not specified
Cell lineMOLT-4

Source evidence

Patent IDCA3215907A1
Compound location

149;149;149

149;149;149 enlarged structure149;149;149 location on patent page 65
Activity table
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