Activity record

PGDB_A068476

Assay: % DegradationTarget: ARQC: ambiguous
Activity overview

degradation = 76 %

TargetAR
Cell lineLNCaP
Concentration7.5 uM
Assay / Readout% Degradation
Assay IDPGDB_AS000627
PatentJP5998117B2
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C026016
Compound IDPGDB_C026016
CompoundASC-JM13
Source record IDPGDB_C026016
InChIKeyQQKDKLCJVCWKBA-HVIAUGEGSA-N

Assay context

Assay IDPGDB_AS000627
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration7.5 uM
Detection targetprotein_degradation
TargetAR
E3Not specified
Cell lineLNCaP
OrganismHomo sapiens

Source evidence

Patent IDJP5998117B2
Compound location

ASC-JM13

ASC-JM13 enlarged structureASC-JM13 location on patent page 63
Activity table
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