PatGlueDB | Molecular Glue Patent Bioactivity Database

Patent summary

Publication numberJP5998117B2

AssigneeAllianz Pharmascience

TitleCompounds with (substituted phenyl) -propenal moieties, derivatives thereof, biological activity and uses thereof

Family ID39609007

Family members28

Filing year2013

Publication date2016-09-28

JurisdictionJP

Compounds13

Activity records50

Assays8

Activity compounds and values

Activity records

50 records

	Control		Value		Concentration	Time				Record ID	Compound	Assay	Details
% Degradation	-	=	48	%	2.5 uM	-	AR	-	LNCaP	PGDB_A007563	PGDB_C026007	PGDB_AS002020	View
% Degradation	-	=	0	%	1 uM	-	AR	-	LNCaP	PGDB_A007766	PGDB_C026017	PGDB_AS002051	View
% Degradation	-	=	7	%	5 uM	-	-	-	CWR22Rv1	PGDB_A007781	PGDB_C026007	PGDB_AS001322	View
% Degradation	-	=	27	%	5 uM	-	AR	-	LNCaP	PGDB_A008995	PGDB_C026008	PGDB_AS002019	View
% Degradation	-	=	23	%	2.5 uM	-	-	-	CWR22Rv1	PGDB_A011123	PGDB_C026014	PGDB_AS002433	View
% Degradation	-	=	11	%	2.5 uM	-	AR	-	LNCaP	PGDB_A011275	PGDB_C026013	PGDB_AS002020	View
% Degradation	-	=	0	%	1 uM	-	AR	-	LNCaP	PGDB_A011482	PGDB_C026006	PGDB_AS002051	View
% Degradation	-	=	0	%	2.5 uM	-	AR	-	LNCaP	PGDB_A012620	PGDB_C026009	PGDB_AS002020	View
% Degradation	-	=	68	%	7.5 uM	-	AR	-	LNCaP	PGDB_A017360	PGDB_C026014	PGDB_AS000627	View
% Degradation	-	=	87	%	7.5 uM	-	-	-	CWR22Rv1	PGDB_A018644	PGDB_C026016	PGDB_AS001947	View
% Degradation	-	=	0	%	2.5 uM	-	AR	-	LNCaP	PGDB_A020127	PGDB_C026016	PGDB_AS002020	View
% Degradation	-	=	29	%	2.5 uM	-	-	-	CWR22Rv1	PGDB_A021795	PGDB_C026015	PGDB_AS002433	View
% Degradation	-	=	15	%	2.5 uM	-	AR	-	LNCaP	PGDB_A022076	PGDB_C026006	PGDB_AS002020	View
% Degradation	-	=	58	%	5 uM	-	AR	-	LNCaP	PGDB_A027804	PGDB_C026011	PGDB_AS002019	View
% Degradation	-	=	50	%	5 uM	-	AR	-	LNCaP	PGDB_A028891	PGDB_C026012	PGDB_AS002019	View
% Degradation	-	=	52	%	7.5 uM	-	AR	-	LNCaP	PGDB_A031547	PGDB_C026009	PGDB_AS000627	View
% Inhibition	-	=	0	%	1 uM	-	-	-	CWR22Rv1	PGDB_A033281	PGDB_C026013	PGDB_AS000637	View
% Degradation	-	=	57	%	2.5 uM	-	-	-	CWR22Rv1	PGDB_A033704	PGDB_C026017	PGDB_AS002433	View
% Degradation	-	=	43	%	5 uM	-	AR	-	LNCaP	PGDB_A033766	PGDB_C026016	PGDB_AS002019	View
% Degradation	-	=	100	%	2.5 uM	-	-	-	CWR22Rv1	PGDB_A035466	PGDB_C026005	PGDB_AS002433	View

Rows per pagePage 1 of 3 · 50 recordsGo to page