Activity record

PGDB_A074229

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

IC50 = 56.2 nM

TargetGSPT1
Cell lineHL-60
Time72 h
Assay / Readoutluminescence / IC50
Assay IDPGDB_AS000799
PatentIL323841A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C008163
Compound IDPGDB_C008163
Compound12
Source record IDPGDB_C008163
InChIKeyAOUHKTNYEATNJX-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000799
Assay familyviability
Assay systemcell_based
ReadoutIC50
Technologyluminescence
Treatment time72 h
Detection target% Cell viability
TargetGSPT1
E3Not specified
Cell lineHL-60

Source evidence

Patent IDIL323841A
Compound location

12

12 enlarged structure12 location on patent page 53
Activity table
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