Activity record

PGDB_A076804

Assay: biochemicalTarget: DCAF15QC: standardized
Activity overview

IC50 <= 10 uM

TargetDCAF15
E3 ligaseDCAF15
Time1 h | <= 1 uM
Assay / ReadoutHTRF / IC50
Assay IDPGDB_AS002163
PatentWO2023059899A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C010006
Compound IDPGDB_C010006
Compound8
Source record IDPGDB_C010006
InChIKeyKBSUAXFXTIHGKS-ZDUSSCGKSA-N

Assay context

Assay IDPGDB_AS002163
Assay familybiochemical
Assay systembiochemical
ReadoutIC50
TechnologyHTRF
Treatment time1 h | <= 1 uM
TargetDCAF15
E3DCAF15

Source evidence

Patent IDWO2023059899A1
Compound location

8

8 enlarged structure8 location on patent page 24
Activity table
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