Activity record

PGDB_A079603

Assay: viabilityTarget: VAV1QC: ambiguous
Activity overview

IC50 = 0.1887 nM

TargetVAV1
Cell linepan-B
Assay / Readoutflow_cytometry / IC50
Assay IDPGDB_AS001016
PatentWO2026051943A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C029558
Compound IDPGDB_C029558
Compound实施例 181
Source record IDPGDB_C029558
InChIKeyGRVXQDQSAQPCQQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001016
Assay familyviability
Assay systemcell_based
ReadoutIC50
Technologyflow_cytometry
TargetVAV1
E3Not specified
Cell linepan-B
OrganismHomo sapiens

Source evidence

Patent IDWO2026051943A1
Compound location

实施例 181

实施例 181 enlarged structure实施例 181 location on patent page 173
Activity table
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