Assay
PGDB_AS000258
System: cell_basedCell line: KG-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.002 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A015133 | PGDB_C001291 | PGDB_AS000258 | View | |
| IC50 | - | = | 0.0015 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A019826 | PGDB_C001288 | PGDB_AS000258 | View | |
| IC50 | - | > | 10 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A024594 | PGDB_C019834 | PGDB_AS000258 | View | |
| IC50 | - | = | 0.001 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A030206 | PGDB_C001290 | PGDB_AS000258 | View | |
| IC50 | - | = | 0.0008 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A033557 | PGDB_C001287 | PGDB_AS000258 | View | |
| IC50 | - | = | 0.0014 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A048219 | PGDB_C001292 | PGDB_AS000258 | View | |
| IC50 | - | > | 10 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A049094 | PGDB_C019833 | PGDB_AS000258 | View | |
| IC50 | - | = | 0.014 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A058207 | PGDB_C001289 | PGDB_AS000258 | View | |
| IC50 | - | = | 4.1 | uM | - | — | - | - | KG-1 | EP4617270A1 | PGDB_A075789 | PGDB_C019835 | PGDB_AS000258 | View |