Assay
PGDB_AS000297
System: biochemicalTarget: CRBN
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.14 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A009862 | PGDB_C025171 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.1 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A016363 | PGDB_C025173 | PGDB_AS000297 | View | |
| IC50 | - | = | 1.43 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A019982 | PGDB_C025168 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.16 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A028393 | PGDB_C025167 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.16 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A037321 | PGDB_C025163 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.05 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A037461 | PGDB_C025170 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.06 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A037892 | PGDB_C025172 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.93 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A038315 | PGDB_C025169 | PGDB_AS000297 | View | |
| IC50 | - | = | 1.57 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A054404 | PGDB_C025164 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.94 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A058026 | PGDB_C025166 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.54 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A058707 | PGDB_C025165 | PGDB_AS000297 | View | |
| IC50 | - | = | 0.25 | uM | - | — | - | - | - | EP3891128A4 | PGDB_A061675 | PGDB_C025164 | PGDB_AS000297 | View |