PatGlueDB | Molecular Glue Patent Bioactivity Database

Assay context summary

Assay context

7 activity records

Assay family% Degradation

Systemcell_based

ReadoutDmax

TargetNEK7

E3CRBN

Cell lineCAL-51

OrganismHomo sapiens

Technologyluminescence

Activity compounds and values

Activity records

7 records

Structure	Metric	Control	Relation	Value	Unit	Concentration	Time	Target	E3	Cell line	Patent	Record ID	Compound	Assay	Details
	Dmax	-	>	75	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A032664	PGDB_C020455	PGDB_AS002252	View
	Dmax	-	>	50	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A032907	PGDB_C020452	PGDB_AS002252	View
	Dmax	-	>	50	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A041672	PGDB_C020453	PGDB_AS002252	View
	Dmax	-	>	50	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A051564	PGDB_C020451	PGDB_AS002252	View
	Dmax	-	>	50	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A055953	PGDB_C020454	PGDB_AS002252	View
	Dmax	-	>	50	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A064090	PGDB_C020450	PGDB_AS002252	View
	Dmax	-	=	79	%	Concentration series: 1 uM, 0.05 nM	24 h	-	-	CAL-51	KR20260041885A	PGDB_A064825	PGDB_C020449	PGDB_AS002252	View

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