Assay

PGDB_AS002533

System: cell_basedTarget: VAV1Cell line: Jurkat
Assay context summary

Assay context

77 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetVAV1
E3Not specified
Cell lineJurkat
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C009181
DC50-=117.365nM-—VAV1-JurkatWO2026013576A1PGDB_A007874PGDB_C009181PGDB_AS002533View
2D structure for PGDB_C009213
DC50-=464.85nM-—VAV1-JurkatWO2026013576A1PGDB_A008135PGDB_C009213PGDB_AS002533View
2D structure for PGDB_C009237
DC50-=81.399nM-—VAV1-JurkatWO2026013576A1PGDB_A008668PGDB_C009237PGDB_AS002533View
2D structure for PGDB_C009180
DC50-=49.892nM-—VAV1-JurkatWO2026013576A1PGDB_A009447PGDB_C009180PGDB_AS002533View
2D structure for PGDB_C009227
DC50-=6873.496nM-—VAV1-JurkatWO2026013576A1PGDB_A010230PGDB_C009227PGDB_AS002533View
2D structure for PGDB_C009203
DC50-=197.593nM-—VAV1-JurkatWO2026013576A1PGDB_A010723PGDB_C009203PGDB_AS002533View
2D structure for PGDB_C009242
DC50-=556.281nM-—VAV1-JurkatWO2026013576A1PGDB_A013420PGDB_C009242PGDB_AS002533View
2D structure for PGDB_C009226
DC50-=9132.535nM-—VAV1-JurkatWO2026013576A1PGDB_A013885PGDB_C009226PGDB_AS002533View
2D structure for PGDB_C009206
DC50-=236.047nM-—VAV1-JurkatWO2026013576A1PGDB_A014104PGDB_C009206PGDB_AS002533View
2D structure for PGDB_C009231
DC50-=10000nM-—VAV1-JurkatWO2026013576A1PGDB_A015981PGDB_C009231PGDB_AS002533View
2D structure for PGDB_C009222
DC50-=2527.218nM-—VAV1-JurkatWO2026013576A1PGDB_A016407PGDB_C009222PGDB_AS002533View
2D structure for PGDB_C009204
DC50-=126.348nM-—VAV1-JurkatWO2026013576A1PGDB_A016459PGDB_C009204PGDB_AS002533View
2D structure for PGDB_C009196
DC50-=97.446nM-—VAV1-JurkatWO2026013576A1PGDB_A016555PGDB_C009196PGDB_AS002533View
2D structure for PGDB_C009169
DC50-=25.757nM-—VAV1-JurkatWO2026013576A1PGDB_A017247PGDB_C009169PGDB_AS002533View
2D structure for PGDB_C009192
DC50-=69.912nM-—VAV1-JurkatWO2026013576A1PGDB_A018972PGDB_C009192PGDB_AS002533View
2D structure for PGDB_C009183
DC50-=86.441nM-—VAV1-JurkatWO2026013576A1PGDB_A019532PGDB_C009183PGDB_AS002533View
2D structure for PGDB_C009182
DC50-=56.303nM-—VAV1-JurkatWO2026013576A1PGDB_A020121PGDB_C009182PGDB_AS002533View
2D structure for PGDB_C009207
DC50-=280.439nM-—VAV1-JurkatWO2026013576A1PGDB_A021305PGDB_C009207PGDB_AS002533View
2D structure for PGDB_C009221
DC50-=2471.921nM-—VAV1-JurkatWO2026013576A1PGDB_A022247PGDB_C009221PGDB_AS002533View
2D structure for PGDB_C009229
DC50-=10000nM-—VAV1-JurkatWO2026013576A1PGDB_A023547PGDB_C009229PGDB_AS002533View
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