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Metrics
| Metric | Activity records | Compounds | Assays | Patents | Units | Details |
|---|---|---|---|---|---|---|
| % Degradation | 20,821 | 7,350 | 236 | 86 | 1 | View |
| IC50 | 19,009 | 9,077 | 764 | 184 | 3 | View |
| DC50 | 12,247 | 7,097 | 276 | 118 | 3 | View |
| EC50 | 8,167 | 4,198 | 114 | 52 | 4 | View |
| Dmax | 7,668 | 4,171 | 188 | 65 | 1 | View |
| % Inhibition | 5,575 | 1,922 | 167 | 32 | 1 | View |
| Emax | 1,096 | 821 | 32 | 11 | 1 | View |
| Ymin | 1,033 | 665 | 10 | 7 | 1 | View |
| GI50 | 984 | 545 | 39 | 14 | 2 | View |
| Kd | 831 | 806 | 24 | 17 | 2 | View |
| Ki | 578 | 461 | 16 | 15 | 2 | View |
| % Cell viability | 380 | 132 | 22 | 10 | 1 | View |
| Selectivity index | 215 | 142 | 8 | 5 | 1 | View |
| ΔTm | 136 | 34 | 4 | 1 | 1 | View |
| Potency ratio | 106 | 75 | 3 | 1 | 1 | View |
| CC50 | 93 | 57 | 13 | 3 | 1 | View |
| Ternary complex response | 55 | 53 | 1 | 1 | 1 | View |
| Fold change | 51 | 49 | 3 | 3 | 1 | View |
| Relative binding | 50 | 25 | 2 | 2 | 1 | View |
| Target engagement | 44 | 22 | 2 | 1 | 1 | View |