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Activity compounds and values
Activity records
| Structure | Metric | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | ||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 2.3 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A000001 | PGDB_C029684 | PGDB_AS001440 | View | |
| DC50 | - | = | 10000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000005 | PGDB_C032272 | PGDB_AS001413 | View | |
| DC50 | - | = | 52 | nM | - | — | IKZF2 | - | Jurkat | WO2026080794A1 | PGDB_A000007 | PGDB_C030846 | PGDB_AS001885 | View | |
| DC50 | - | = | 10000 | nM | - | — | SMARCA4 | - | Calu-6 | WO2026128580A1 | PGDB_A000008 | PGDB_C032265 | PGDB_AS001413 | View | |
| DC50 | - | = | 5 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A000016 | PGDB_C029462 | PGDB_AS001440 | View | |
| DC50 | - | = | 92 | nM | - | — | IKZF1 | - | Jurkat | WO2026080794A1 | PGDB_A000023 | PGDB_C030999 | PGDB_AS000302 | View | |
| DC50 | - | = | 2 | nM | - | — | VAV1 | - | - | WO2026119120A1 | PGDB_A000026 | PGDB_C032005 | PGDB_AS001984 | View |